Browsing Sivas Teknik Bilimler Meslek Yüksekokulu by Author "https://orcid.org/0000-0002-0420-2043"
Now showing items 1-15 of 15
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1,2,3-Triazole substituted phthalocyanine metal complexes as potential inhibitors for anticholinesterase and antidiabetic enzymes with molecular docking studies
Koçyiğit, Ümit M.; Taslimi, Parham; Tüzün,Burak; Yakan, Hasan; Muğlu, Halit; Güzel, Emre (09.12.2020)In recent years, acetylcholinesterase (AChE) and a-glycosidase (a-gly) inhibition have emerged as a promising and important approach for pharmacological intervention in many diseases such as glaucoma, epilepsy, obesity, ... -
Architectural View of Flexible Aliphatic –OH Group Coordinated Hemi‑Directed Pb(II)‑Salen Coordination Polymer: Synthesis, Crystal Structure, Spectroscopic Insights, Supramolecular Topographies, and DFT Perspective
Majumdar, Dhrubajyoti; Tüzün,Burak; Pal, Tapan Kumar; Das, Sourav; Bankura, Kalipada (27.01.2022, 27.01.2022)We serendipitously designed one novel 1D hetero-binuclear Zn(II)-Pb(II) coordination polymer, namely [(Zn)(Pb)(L)(η1– NCS)(η1–SCN)]n (1) from Salen ligand ( H3L) in the presence of NaSCN. The complex was structurally ... -
Benzotriazole-oxadiazole hybrid Compounds: Synthesis, anticancer Activity, molecular docking and ADME profiling studies
Mermer, Arif; Bulbul, Muhammet Volkan; Kalender, Semiha Mervenur; Keskin, Ilknur; Tuzun, Burak; Eyupoglu, Ozan Emre (29.04.2022)Herein the designed novel benzotriazole-oxadiazole hybrid compounds were synthesized using both conventional method and ultrasound sonication (US) as an environmentally friendly method. It was observed that the US method ... -
Biological effects and molecular docking studies of Catechin 5-O-gallate: antioxidant, anticholinergics, antiepileptic and antidiabetic potentials
Taslimi, Parham; Kocyigit, Umit M.; Tüzün,Burak; Kirici, Mahinur (Journal of Biomolecular Structure and Dynamics, 04.10.2020)Gallocatechin gallate is a form of catechin and an ester of gallocatechin and gallic acid. This is an epimer of the gallate epigallocatechin. In this study, the effect of this molecule, containing a biologically active ... -
Biosorption of Rhodamine B dye from aqueous solution by Rhus coriaria L. plant: Equilibrium, kinetic, thermodynamic and DFT calculations
Celik, Muhammed Safa; Cetinus, Senay Akkus; Yenidunya, Ali Fazıl; Cetinkaya, Serap; Tüzün,Burak (Journal of Molecular Structure, 16 Septemb)Water-soluble basic rhodamine B (RhB) was adsorbed onto fruit powders of Rhus coriaria L. (Anacar- diaceae), sumac in batch reactions. Adsorption was optimized by employing concentration, pH, and time parameters. Experimental ... -
Corrosion inhibition of Carbon Steel using a new morpholine-based ligand during acid pickling: Experimental and theoretical studies
Rezaeivala, Majid; Bozorg, Mansoor; Rafiee, Negar; Sayin, Koray; Tuzun, Burak (Inorganic Chemistry Communications, 12 Decembe)Here, a novel, relatively inexpensive Schiff base ligand (HL) has been studied as a corrosion inhibitor for the protection of steel in acidic solution. Different concentrations (0–25 ppm) of HL were added to the test ... -
Eco-friendly and potential colin esterase enzyme inhibitor agent sulfonyl hydrazone series: Synthesis, Bioactivity Screening, DFT, ADME properties, and Molecular Docking study
Ozmen, Ummuhan Ozdemir; Tuzun, Burak; Ayan, Esra Bilen; Cevrimli, Bekir Sıtkı (Journal of Molecular Structure, 4 April 20)In this study, new compounds containing the sulfonamide group and having inhibitory activity on cholinesterase enzymes (AChE, BChE) were synthesized. For this purpose, three new sulfonylhydrazone compounds were synthesized ... -
Experimental and computational investigation of 3,5-di-tert-butyl-2-(((3-((2-morpholinoethyl)(pyridin-2-ylmethyl) amino) propyl)imino) methyl)phenol and related reduced form as an inhibitor for C-steel
Karimi, Saeid; Rezaeivala, Majid; Sayin, Koray; tüzün, burak (16.04.2022)The effect of new compounds containing morpholine moiety including: 3,5-di-tert-butyl-2-(((3-((2-morpholinoethyl)( pyridine-2-ylmethyl)amino)propyl)imino)methyl)phenol (L1) and its reduced form, 3,5-di-tert-butyl-2-(((3 ... -
Experimental and theoretical investigation of corrosion inhibition effect of two piperazine-based ligands on carbon steel in acidic media
Rezaeivala, Majid; Karimi, Saeid; Sayin, Koray; Tüzün,Burak (4.02.2022)hydroxyethyliminomethyl) phenyl)piperazine (1) or its reduced form, 1,4-bis(2-(2-hydroxyethylaminomethyl)phenyl)piperazine (2), as possible corrosion inhibitors, were compared to a solution containing no (1) or (2). The ... -
In vitro cytotoxic effects, in silico studies, some metabolic enzymes inhibition, and vibrational spectral analysis of novel β-amino alcohol compounds
Tas, Ayca; Tüzün,Burak; Ali, N.; Taslimi, Parham; Agbektas, Tugba; Cakmak, Nese Keklikcioglu (Journal of Molecular Structure, 8 October )In this study, an efficient single-step method for the preparation of β-amino alcohols ( 1 –3 ) in aqueous media was applied. The aim was to investigate the cytotoxic activity of Compounds 1, 2 and 3 in neu- roblastoma ... -
Moderate DNA and high SARS-CoV-2 spike protein affinity of oxidovanadium(IV) complexes of 2-furoic acid hydrazones: In silico and in vitro approach
Zahirovi, Adnan; Tüzün,Burak; Hadzalic, Selma; Osmankovic, Irnesa; Roca, Suncica; Begic, Sabina; Focak, Muhamed (Journal of Molecular Structure, 1 Septembe)The interaction of five neutral heteroleptic octahedral paramagnetic mononuclear oxidovanadium(IV) complexes of general composition [VIVO(bpy)L], where L is a dianionic tridentate ONO-donor hydrazone ligand derived from ... -
Quinoline-fused both non-peripheral and peripheral ZnII and MgII phthalocyanines: Anti-cholinesterase, anti- α-glucosidase, DNA nuclease, antioxidant activities, and in silico studies
Yalazan, Halise; Tüzün,Burak; Akkaya, Didem; Barut, Burak; Kantekin, Halit; Yıldırmıs, Sermet (08.04.2022)Quinoline-fused ZnII (ZnPcp/ZnPcnp) and MgII (MgPcp/MgPcnp) phthalocyanines with four 4-methylquinolin-2-ol (1) at non-peripheral or peripheral positions of the phthalocyanine core have been synthesized via cyclotetramerization ... -
Repositioning of acefylline as anti-cancer drug: Synthesis, anticancer and computational studies of azomethines derived from acefylline tethered 4-amino-3- mercapto-1,2,4-triazole
Shahzadi, Irum; Zahoor, Ameer Fawad; Tüzün,Burak; Mansha, Asim; Anjum, Muhammad Naveed; Rasul, Azhar; Irfan, Ali; Kotwica-Mojzych, Katarzyna; Mojzych, Mariusz (PLOS ONE, 15.12.2022)Novel azomethines derived from acefylline tethered triazole hybrids (7a-k) have been synthesized and evaluated against human liver cancer cell line (Hep G2) using MTT assay. The synthesized series of azomethines exhibited ... -
Synthesis, characterization, crystallographic aspects, Fukui function, and photodynamic antifungal chemotherapy investigation of Cd (II)-tricyanomethanide coordination polymer: Insights from DFT
Majumdar, Dhrubajyoti; Philip, Jessica Elizabeth; Tüzün,Burak; Roy, Sourav (Inorganic Chemistry Communications, 8 July 202)This study delves into the synthesis, crystal structure, structural topology, photodynamic antifungal therapy (PACT), and DFT-based investigations of one [Cd(TCM)2]n coordination polymer (TCM = tricyanomethanide). The ... -
Unravelling the Synthetic Mimic, Spectroscopic Insights, and Supramolecular Crystal Engineering of an Innovative Heteronuclear Pb(II)‑Salen Cocrystal: An Integrated DFT, QTAIM/NCI Plot, NLO, Molecular Docking/PLIP, and Antibacterial Appraisal
Majumdar, Dhrubajyoti; Philip, Jessica Elizabeth; Tüzün,Burak; Frontera, A.; Gomila, Rosa M.; Roy, Sourav; Bankura, Kalipada (springer, 26.07.2022)Spontaneous self-assembly in the supramolecular entity is one of the enthralling synthetic routes. It produces disparate structure crystal complexes after selecting suitable M-L combinations in the pseudohalide sense. In ...